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View a video* illustrating
Fampridine-SR’s mechanism of action:
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Researchers have shown that, contrary to popular
belief, most people with spinal cord injury (SCI) do not
have severed cords; rather, most have blunt damage to
the cord. The great majority of such individuals have
some axons within the spinal cord that survive the
injury. However, these surviving axons often are damaged
and lose part of their myelin, the insulating sheath
that permits electrical impulses to be conducted down
the axon. Nerve impulses "short circuit" in demyelinated
axons, much like electricity in a wire whose insulation
is stripped. Thus, even though a demyelinated axon is
alive, it cannot transmit motor or sensory impulses. In
multiple sclerosis (MS), the myelin is believed to be
damaged by the body's own immune system, rather than by
physical trauma as in SCI.

Fampridine-SR's major action is to block specialized potassium channels on axons. When an axon is demyelinated after injury, large numbers of these potassium channels are exposed and "leak" potassium ions, causing the axon to "short circuit".

By closing the exposed potassium channels, Fampridine-SR permits the axon to transmit impulses again, even in a demyelinated state.
View a video* illustrating
Fampridine-SR’s mechanism of action:
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(4.0MB) Small
(2.8MB)
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